Oxidative alpha,omega-diyne coupling as an approach towards novel peptidic macrocycles.
Verlinden, S.; Geudens, N.; Martins, J. C.; Tourwe, D.; Ballet, S.; Verniest, G., Org. Biomol. Chem. 2015, 13, 9398-9404.
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Suzuki-Miyaura Diversification of Amino Acids and Dipeptides in Aqueous Media.
Willemse, T.; Van Imp, K.; Goss, R. J. M.; Van Vlijmen, H. W. T.; Schepens, W.; Maes, B. U. W.; Ballet, S., ChemCatChem 2015, 7, 2055-2070.
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Homohalocyclization: Electrophilic Bromine-Induced Cyclizations of Cyclopropanes
C. Rösner, U. Hennecke, Org. Lett. 2015, 17, 3226-3229.
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Synthesis and biological evaluation of compact, conformationally constrained bifunctional opioid agonist – Neurokinin-1 antagonist peptidomimetics.
Guillemyn, K.; Kleczkowska, P.; Lesniak, A.; Dyniewicz, J.; Van der Poorten, O.; Van den Eynde, I.; Keresztes, A.; Varga, E.; Lai, J.; Porreca, F.; Chung, N. N.; Lemieux, C.; Mika, J.; Rojewska, E.; Makuch, W.; Van Duppen, J.; Przewlocka, B.; Vanden Broeck, J.; Lipkowski, A. W.; Schiller, P.
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Structural basis for bifunctional peptide recognition at human delta-opioid receptor.
Fenalti, G.; Zatsepin, N. A.; Betti, C.; Giguere, P.; Han, G. W.; Ishchenko, A.; Liu, W.; Guillemyn, K.; Zhang, H.; James, D.; Wang, D.; Weierstall, U.; Spence, J. C. H.; Boutet, S.; Messerschmidt, M.; Williams, G. J.; Gati, C.; Yefanov, O. M.; White, T. A.; Oberthuer, D.; Metz, M.; Yoon, C.
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Iodoalkanes: Synthesis by Addition to π-Type C-C-Bonds (Update 2014)
U. Hennecke in Science of Synthesis Knowledge Updates 2015/2, T. Wirth (Ed.), Thieme, Stuttgart, 2015, 437-448.
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Rational design of a hexapeptide hydrogelator for controlled-release drug delivery.
Bibian, M.; Mangelschots, J.; Gardiner, J.; Waddington, L.; Diaz Acevedo, M. M.; De Geest, B. G.; Van Mele, B.; Madder, A.; Hoogenboom, R.; Ballet, S., J. Mater. Chem. B 2015, 3, 759-765.
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Asymmetric, Organocatalytic Bromolactonization of Allenoic Acids
M. Wilking, C. G. Daniliuc, U. Hennecke, Synlett 2014, 25, 1701-1704.
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Draft genome sequence analysis of a Pseudomonas putida W15Oct28 strain with antagonistic activity to Gram-positive and Pseudomonas sp. pathogens.
Ye, L. M.; Hildebrand, F.; Dingemans, J.; Ballet, S.; Laus, G.; Matthijs, S.; Berendsen, R.; Cornelis, P., Plos One 2014, 9, e110038
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Silaproline Helical Mimetics Selectively Form an All-trans PPII Helix.
Martin, C.; Legrand, B.; Lebrun, A.; Berthomieu, D.; Martinez, J.; Cavelier, F., Eur. Chem. J. 2014, 20, 14240-14244.
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Rational Design of Injectable Hexapeptide Hydrogelators for Controlled-Release Drug Delivery.
Bibian, M.; Mangelschots, J.; Martin, C.; Gardiner, J.; Waddington, L.; Acevedo, M. M. D.; Van Mele, B.; Madder, A.; Hoogenboom, R.; Ballet, S., J. Pept. Sci. 2014, 20, S208-S208
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Efficient synthesis of conformationally constrained, amino-triazoloazepinone-containing di- and tripeptides via a one-pot Ugi-Huisgen tandem reaction.
Barlow, T. M. A.; Jida, M.; Tourwe, D.; Ballet, S., Org. Biomol. Chem. 2014, 12, 6986-6989.
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